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Products Details
Product Description
– LSD1-IN-22 is a potent Lysine-specific demethylase 1 (LSD1) inhibitor with a Ki value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells[1].
Web ID
– HY-151191
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C9H8BrF2N
References
– [1]Hideaki Niwa, et al. Structure-Activity Relationship and In Silico Evaluation of cis- and trans-PCPA-Derived Inhibitors of LSD1 and LSD2. ACS Medicinal Chemistry Letters Article ASAP.
CAS Number
– 2821068-05-5
Molecular Weight
– 248.07
SMILES
– N[C@H]1[C@H](C2=CC(F)=C(Br)C=C2F)C1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Demethylase
Isoform
– KDM1/LSD1
Pathway
– Epigenetics
Product type
– Reference compound
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