SGC2085 HCl
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SGC2085 HCl

SKU T4013-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 136 CAD through 1,904 CAD

Products Details

Product Description

– SGC2085 is a potent and selective coactivator associated arginine methyltransferase 1 (CARM1) Inhibitor with an IC50 of 50 nM and more than undred-fold selectivity over other PRMTs. CARM1 is an important positive modulator of Wnt/β-catenin transcription and neoplastic transformation in colorectal cancer as well as a critical factor in estrogen-stimulated breast cancer growth, and its depletion results in decreased proliferation of myeloid leukemia cells in vivo.

Web ID

– T4013

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C19H24N2O2·HCl

References

– Renato., et al. Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening . J Med Chem. 2016 Jul 28;59(14):6838-47.

CAS Number

– 1821908-49-9

Molecular Weight

– C19H24N2O2·HCl

Compound Purity

– 0.9991

SMILES

– C(=O)([C@H](C)N)NCc1cc(c(cc1)Oc1cc(cc(c1)C)C)C.Cl

Pathway

– Chromatin/Epigenetic

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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