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PF-05381941

SKU T36017-1 mL * 10 mM (in DMSO) Category Small Compound Brand: TargetMol

Price range: 144 CAD through 1,139 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

1 mg 1 mL * 10 mM (in DMSO)10 mg 25 mg 5 mg

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Products Details

Product Description

– PF-05381941 is a selective and potent dual inhibitor of TAK1 and p38α with IC 50 =156 nM/186nM that inhibits the kinase activity of TAK1 by binding to its active site.

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T36017

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C27H26N6O2

References

– Kilty I, et al. TAK1 inhibition in the DFG-out conformation. Chem Biol Drug Des. 2013;82(5):500-505.

CAS Number

– 1474022-02-0

Molecular Weight

– C27H26N6O2

Compound Purity

– 0.9804

SMILES

– N#CC1=CC=CC(=C1)N2N=C(C=C2NC(=O)NC3=CC=C(OC=4C=CN=CC4)C(=C3)C)C(C)(C)C

Pathway

– MAPK

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.