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SR 16832

SKU T24827-5 mg Category Small Compound Brand: TargetMol

Price range: 61 CAD through 734 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

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Products Details

Product Description

– SR 16832 is a dual-site PPARγ inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPARγ, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T24827

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C17H12ClN3O4

References

– Brust et al (2017) Modification of the othosteric PPARγ covalent antagonist scaffold yields an improved dual-site allosteric inhibitor. ACS Chem.Biol. 12 969

CAS Number

– 2088135-12-8

Molecular Weight

– C17H12ClN3O4

Compound Purity

– 0.9996

SMILES

– N(C(=O)C1=CC(N(=O)=O)=CC=C1Cl)C=2C3=C(C=CC(OC)=C3)N=CC2

Pathway

– DNA Damage/DNA Repair|||Metabolism

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.