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GSK699

SKU T32010-1 mg Category PROTAC Brand: TargetMol

Price range: 2,720 CAD through 5,280 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

1 mg 10 mg 25 mg 5 mg 50 mg

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Products Details

Product Description

– GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T32010

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C45H51BrN8O7

References

– Bassi ZI, Fillmore MC, Miah AH, Chapman TD, Maller C, Roberts EJ, Davis LC, Lewis DE, Galwey NW, Waddington KE, Parravicini V, Macmillan-Jones AL, Gongora C, Humphreys PG, Churcher I, Prinjha RK, Tough DF. Modulating PCAF/GCN5 Immune Cell Function through a PROTAC Approach. ACS Chem Biol. 2018 Oct 19;13(10):2862-2867. doi: 10.1021/acschembio.8b00705. Epub 2018 Sep 18. PubMed PMID: 30200762.

CAS Number

– 2260944-68-9

Molecular Weight

– C45H51BrN8O7

SMILES

– O=C1C=2C(C(=O)N1C3C(=O)NC(=O)CC3)=CC=CC2OCCCC4=CC=C(N(CCCN(C(=O)C5=CC=C(C=C5)[C@H]6C[C@@H](NC7=C(Br)C(=O)N(C)N=C7)CN(C)C6)C)C)C=C4

Target

– Apoptosis|||Caspase|||HIV Protease|||AMPK

Pathway

– Others

Product type

– PROTAC

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.