Download Files:

bio-THZ1

SKU T10546-10 mg Category Small Compound Brand: TargetMol

Price range: 3,677 CAD through 7,536 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

10 mg 25 mg

Clear

Products Details

Product Description

– bio-THZ1 is a biotinylated version of THZ1, a selective and irreversibly covalent CDK7 inhibitor (IC50: 3.2 nM).

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T10546

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C52H65ClN12O8S

References

– Kwiatkowski N, et al. Targeting transcription regulation in cancer with a covalent CDK7 inhibitor. Nature. 2014 Jul 31;511(7511):616-20.

CAS Number

– 1604811-14-4

Molecular Weight

– C52H65ClN12O8S

SMILES

– [H][C@]12CS[C@@H](CCCCC(=O)NCCOCCOCCOCCNC(=O)NCCCN(C)CC=CC(=O)Nc3ccc(cc3)C(=O)Nc3cccc(Nc4ncc(Cl)c(n4)-c4c[nH]c5ccccc45)c3)[C@@]1([H])NC(=O)N2

Target

– Adrenergic Receptor|||Endogenous Metabolite

Pathway

– Cell Cycle/Checkpoint

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.