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AZ’3137
For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.
Products Details
Product Description
– AZ’3137 (Compound 22) is an orally active PROTAC-based androgen receptor (AR) degrader, exhibiting a DC50 value of 22 nM. It inhibits cell proliferation in LNCaP cells with a GI50 of 74 nM. Additionally, AZ’3137 suppresses AR signaling and tumor growth in a prostate cancer mouse model.
For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.
Web ID
– T89238
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C43H47F4N7O4
CAS Number
– 2960179-55-7
Molecular Weight
– C43H47F4N7O4
SMILES
– N#CC1=CC=C(C(F)=C1C(F)(F)F)N2CCC(C3=CC=C(C=C3)N4CCC(CN5CCN(C6=CC(OC)=C7C(=O)N(CC7=C6)C8C(=O)NC(=O)CC8)CC5)CC4)CC2
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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