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ERK5-IN-2

SKU T5535-1 mL * 10 mM (in DMSO) Category Small Compound Brand: TargetMol

Price range: 66 CAD through 1,419 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

1 mg 1 mL * 10 mM (in DMSO)10 mg 100 mg 200 mg 25 mg 5 mg 50 mg

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Products Details

Product Description

– ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50 values of 0.82 μM for ERK5 and 3 μM for ERK5 (MEF2D).

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T5535

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C17H11BrFN3O2

References

– Myers SM, Miller DC, Molyneux L, et al .Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38α and BRD4[J].Eur J Med Chem. 2019 Sep 15;178:530-543.

CAS Number

– 1888305-96-1

Molecular Weight

– C17H11BrFN3O2

Compound Purity

– ≥95%

SMILES

– Fc1cccc(Br)c1C(=O)c1c[nH]c(c1)C(=O)Nc1cccnc1

Pathway

– MAPK

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.