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GAT211
Price range: 48 CAD through 1,333 CAD
Products Details
Product Description
– GAT211 (AZ-4) is a selective and potent cannabinoid 1 receptor (CB1R) orthosteric modulator (PAM) with high affinity for cAMP and β-arrestin2.GAT211 has IOP-lowering and antipsychotic effects and can be used in the study of epilepsy.
Web ID
– T27405
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C22H18N2O2
References
– Garai S, et al. Design, synthesis, and pharmacological profiling of cannabinoid 1 receptor allosteric modulators: Preclinical efficacy of C2-group GAT211 congeners for reducing intraocular pressure. Bioorg Med Chem. 2021 Nov 15;50:116421.
CAS Number
– 102704-40-5
Molecular Weight
– C22H18N2O2
Compound Purity
– 0.997
SMILES
– [O-][N+](=O)CC(c1c([nH]c2ccccc12)-c1ccccc1)c1ccccc1
Pathway
– GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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