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Omarigliptin

SKU T2316-1 mL * 10 mM (in DMSO) Category Small Compound Brand: TargetMol

Price range: 54 CAD through 1,888 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

2 mg 1 mg 1 mL * 10 mM (in DMSO)10 mg 100 mg 25 mg 5 mg 50 mg 500 mg

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Products Details

Product Description

– Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. [3]

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T2316

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C17H20F2N4O3S

Citations

– 1. Du H, Wang S Omarigliptin Mitigates Lipopolysaccharide-Induced Neuroinflammation and Dysfunction of the Integrity of the Blood–Brain Barrier. ACS Chemical Neuroscience. 2020 2. Heo R, Kang M, Mun S Y, et al. Antidiabetic Omarigliptin Dilates Rabbit Aorta by Activating Kv Channels and the SERCA Pump. Fundamental & Clinical Pharmacology. 2022 3. Heo R, Kang M, Mun S Y, et al.Antidiabetic omarigliptin dilates rabbit aorta by activating voltage‐dependent K+ channels and the sarco/endoplasmic reticulum Ca2+‐ATPase pump.Fundamental & Clinical Pharmacology.2023, 37(1): 75-84.

References

– Biftu T, et al. J Med Chem. 2014 Apr 24;57(8):3205-12.

CAS Number

– 1226781-44-7

Molecular Weight

– C17H20F2N4O3S

Compound Purity

– 0.9977

SMILES

– CS(=O)(=O)n1cc2CN(Cc2n1)[C@H]1CO[C@@H]([C@@H](N)C1)c1cc(F)ccc1F

Pathway

– Proteases/Proteasome|||Ubiquitination

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.