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Products Details
Product Description
– BRD4-IN-2 is a bromodomain BRD4 inhibitor with an IC50 value of 9.9 nM.
Web ID
– HY-141843
Shipping
– Room temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C43H48N8O11
References
– [1]Sabnis RW. Substituted 2,3-Benzodiazepines Derivatives as Bromodomain BRD4 Inhibitors. ACS Med Chem Lett. 2021 Sep 28;12(10):1530-1531.
CAS Number
– 2679925-55-2
Molecular Weight
– 852.89
SMILES
– CNC(N1N=C(C2=C(C[C@@H]1C)C=C(C(OC)=C2)OC)C3=CC=C(C=C3)N4CCN(CC4)C(COCCOCC(NC5=C6C(N(C(C6=CC=C5)=O)C7CCC(NC7=O)=O)=O)=O)=O)=O
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
