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Telcagepant

Name: Telcagepant | Agonist — Buy Online | Immunomart
Brand: TargetMol
SKU: T16093-1 mg
Price: 139 CAD
Availability: InStock

SKU T16093-1 mg Category Small Compound Brand: TargetMol

139 CAD

Only 1000 item(s) left in stock.

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Products Details

Product Description

– Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors and reduces neurotransmission in the central nervous system and is used in the study of migraines and for pain relief.

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T16093

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C26H27F5N6O3

References

– Salvatore CA, et al. Pharmacological characterization of MK-0974 [N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-trifluoroethyl)azepan-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide], a potent and orally active calcitonin gene-related peptide receptor antagonist for the treatment of migraine. J Pharmacol Exp Ther. 2008 Feb;324(2):416-21. Epub 2007 Nov 26.

CAS Number

– 781649-09-0

Molecular Weight

– C26H27F5N6O3

Compound Purity

– 0.9898

SMILES

– O=C1N(C=2C(N1)=NC=CC2)C3CCN(C(N[C@H]4C(=O)N(CC(F)(F)F)C[C@@H](CC4)C5=C(F)C(F)=CC=C5)=O)CC3

Target

– Others

Pathway

– GPCR/G Protein|||Neuroscience

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.