GSK3368715
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GSK3368715

SKU T11500-25 mg Category Brand:

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Products Details

Product Description

– GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). It has strong anti-cancer activity.

Web ID

– T11500

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C20H38N4O2

References

– Fedoriw A, et al. Anti-tumor Activity of the Type I PRMT Inhibitor, GSK3368715, Synergizes with PRMT5 Inhibition through MTAP Loss. Cancer Cell. 2019 Jul 8;36(1):100-114.e25.

CAS Number

– 1629013-22-4

Molecular Weight

– C20H38N4O2

SMILES

– C(OCC)C1(COCC)CCC(CC1)C=2C(CN(CCNC)C)=CNN2

Target

– HIV Protease

Pathway

– Chromatin/Epigenetic

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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