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GSK2973980A

SKU T11491-25 mg Category Small Compound Brand: TargetMol

Price range: 3,152 CAD through 5,440 CAD

For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.For sale to research organizations and laboratories only; not for patients or for personal use.

Size

100 mg 25 mg 50 mg

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Products Details

Product Description

– GSK2973980A is a selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor (IC50: 3 nM).

For Research Use Only (RUO). This product is sold strictly for laboratory research use only. Not for human or veterinary consumption, therapeutic, or diagnostic use. Any pharmacological, therapeutic, cosmetic, or biological effects described above are provided as research context only and do not represent intended or approved uses of this product.

Web ID

– T11491

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C25H19F5N4O4

References

– Cheung M, et al. Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1. ACS Med Chem Lett. 2018 Jan 16;9(2):103-108.

CAS Number

– 2219321-25-0

Molecular Weight

– C25H19F5N4O4

SMILES

– C(C(F)(F)F)[C@]1(CC(O)=O)C(=O)C=2C(CC1)=CC(=CC2)C=3C=NC(NC(NC4=CC(F)=C(F)C=C4)=O)=CN3

Target

– Amino Acids and Derivatives

Pathway

– Metabolism

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.