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ESI-08
Price range: 82 CAD through 728 CAD
Products Details
Product Description
– ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.
Web ID
– T11234
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C20H23N3OS
References
– Chen H, et al. 5-Cyano-6-oxo-1,6-dihydro-pyrimidines as potent antagonists targeting exchange proteins directly activated by cAMP. Bioorg Med Chem Lett. 2012 Jun 15;22(12):4038-43.
CAS Number
– 301177-43-5
Molecular Weight
– C20H23N3OS
Compound Purity
– 0.9905
SMILES
– Cc1ccc(C)c(CSc2nc(C3CCCCC3)c(C#N)c(=O)[nH]2)c1
Target
– CDK
Pathway
– GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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