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ERK1/2 inhibitor 1
Price range: 205 CAD through 2,080 CAD
Products Details
Product Description
– ERK1/2 inhibitor 1 is a potent, orally bioavailable compound that exhibits 60% inhibition at 1 nM and has an IC50 of 3.0 nM against ERK1 and ERK2, respectively.
Web ID
– T11226
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C29H32ClN5O4
References
– Heightman TD, et al. Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. J Med Chem. 2018 Jun 14;61(11):4978-4992.
CAS Number
– 2095719-90-5
Molecular Weight
– C29H32ClN5O4
Compound Purity
– 0.9909
SMILES
– C[C@@H](N1Cc2ccc(cc2C1=O)-c1nc(NC2CCOCC2)ncc1Cl)C(=O)N[C@H](CO)c1cccc(C)c1
Target
– DNA/RNA Synthesis
Pathway
– MAPK
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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