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BET-IN-6
Price range: 2,432 CAD through 4,000 CAD
Products Details
Product Description
– BET-IN-6, a ligand with potent and high affinity for inhibiting BRD2/BRD4, plays a crucial role in the synthesis of PROTAC BRD2/BRD4 degrader-1 [1], targeting the protein BRD2/4.
Web ID
– T10522
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C22H20N2O6S
References
– Jiang F, et al. Discovery of novel small molecule induced selective degradation of the bromodomain and extra-terminal (BET) bromodomain protein BRD4 and BRD2 with cellular potencies.Bioorg Med Chem. 2020 Jan 1;28(1):115181.
CAS Number
– 2570470-39-0
Molecular Weight
– C22H20N2O6S
SMILES
– N(S(=O)(=O)C1=C(OC)C=CC=C1)C=2C=3C4=C(C=C(CCC(O)=O)C3)C(=O)N(C)C4=CC2
Target
– 5-HT Receptor|||CCR
Pathway
– Chromatin/Epigenetic
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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