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Products Details
Product Description
– SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.
Web ID
– T203513
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C27H34N4O2
CAS Number
– 1849603-79-7
Molecular Weight
– C27H34N4O2
SMILES
– OCCN(C=1C=CC=2N=C(N=C(C2C1)N3CCC(C=4C=CC=CC4OC)CC3)C5(C)CC5)C
Target
– PI3K
Pathway
– GPCR/G Protein
Product type
– Small Compound
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