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Products Details
Product Description
– PITCOIN4 is a highly selective Class II Alpha PI3K-C2α inhibitor. PITCOIN4 shows nanomolar inhibition of PI3K-C2α and >100-fold selectivity in a general kinase panel[1].
Web ID
– HY-156406
Shipping
– Room temperature
Molecular Formula
– C30H29N7O3S2
References
– [1]Murat Kücükdisli, et al. Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition. J Med Chem. 2023 Oct 26;66(20):14278-14302.
Molecular Weight
– 599.73
SMILES
– CC(C)(NC(CC1=CSC(NC(CSC(N2CCC3=CC=CC=C3)=NC4=C(C2=O)N=CC=N4)=O)=N1)=O)C5=CC=CC=C5
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– 10 mM in DMSO
Target
– PI3K
Pathway
– PI3K/Akt/mTOR
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
