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Products Details
Product Description
– LSD1-IN-22 is a potent Lysine-specific demethylase 1 (LSD1) inhibitor with a Ki value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells[1].
Web ID
– HY-151191
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C9H8BrF2N
References
– [1]Hideaki Niwa, et al. Structure-Activity Relationship and In Silico Evaluation of cis- and trans-PCPA-Derived Inhibitors of LSD1 and LSD2. ACS Medicinal Chemistry Letters Article ASAP.
CAS Number
– 2821068-05-5
Molecular Weight
– 248.07
SMILES
– N[C@H]1[C@H](C2=CC(F)=C(Br)C=C2F)C1
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Demethylase
Isoform
– KDM1/LSD1
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
