Products Details

Product Description

– GPR88 agonist 2 (compound 53) is a potent and brain-penetrantGPR88 agonist with an EC50 value of 14 µM in GPR88 cAMP functional assay[1].

Web ID

– HY-156772

Shipping

– Room temperature

Molecular Formula

– C26H33N5O3

References

– [1]Rahman MT, et al. Evaluation of Amide Bioisosteres Leading to 1,2,3-Triazole Containing Compounds as GPR88 Agonists: Design, Synthesis, and Structure-Activity Relationship Studies. J Med Chem. 2021 Aug 26;64(16):12397-12413.

CAS Number

– 2821859-71-4

Molecular Weight

– 463.57

SMILES

– CNC(C(N=N1)=CN1C[C@@H](C2=CC=C(C=C2)OC[C@@H](C)CC)NC([C@H](C3=CC=CC=C3)C)=O)=O

Clinical Information

– No Development Reported

Research Area

– Neurological Disease; Others

Solubility

– 10 mM in DMSO

Target

– GPR88

Pathway

– GPCR/G Protein

Product type

– Reference compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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