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GPR88 agonist 2
SKU
HY-156772-Get quote
Category Reference compound
Tags GPCR/G Protein, GPR88, Neurological Disease; Others
Products Details
Product Description
– GPR88 agonist 2 (compound 53) is a potent and brain-penetrantGPR88 agonist with an EC50 value of 14 µM in GPR88 cAMP functional assay[1].
Web ID
– HY-156772
Shipping
– Room temperature
Molecular Formula
– C26H33N5O3
References
– [1]Rahman MT, et al. Evaluation of Amide Bioisosteres Leading to 1,2,3-Triazole Containing Compounds as GPR88 Agonists: Design, Synthesis, and Structure-Activity Relationship Studies. J Med Chem. 2021 Aug 26;64(16):12397-12413.
CAS Number
– 2821859-71-4
Molecular Weight
– 463.57
SMILES
– CNC(C(N=N1)=CN1C[C@@H](C2=CC=C(C=C2)OC[C@@H](C)CC)NC([C@H](C3=CC=CC=C3)C)=O)=O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease; Others
Solubility
– 10 mM in DMSO
Target
– GPR88
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.