GAT211

SKU T27405-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 48 CAD through 1,333 CAD

Products Details

Product Description

– GAT211 (AZ-4) is a selective and potent cannabinoid 1 receptor (CB1R) orthosteric modulator (PAM) with high affinity for cAMP and β-arrestin2.GAT211 has IOP-lowering and antipsychotic effects and can be used in the study of epilepsy.

Web ID

– T27405

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C22H18N2O2

References

– Garai S, et al. Design, synthesis, and pharmacological profiling of cannabinoid 1 receptor allosteric modulators: Preclinical efficacy of C2-group GAT211 congeners for reducing intraocular pressure. Bioorg Med Chem. 2021 Nov 15;50:116421.

CAS Number

– 102704-40-5

Molecular Weight

– C22H18N2O2

Compound Purity

– 0.997

SMILES

– [O-][N+](=O)CC(c1c([nH]c2ccccc12)-c1ccccc1)c1ccccc1

Pathway

– GPCR/G Protein

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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