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Product Description
– ERK5-IN-6 (compound 5J) is an ERK5 kinase inhibitor with anticancer activity. ERK5-IN-6 exhibits good anti-proliferative activity with the IC50 value of 4.56 µg/mL for A549 cells[1].
Web ID
– HY-156451
Shipping
– Room temperature
Molecular Formula
– C23H21N3
References
– [1]Qin Zhang, et al. Design, synthesis and SAR of novel 7-azaindole derivatives as potential Erk5 kinase inhibitor with anticancer activity. Bioorg Med Chem. 2023 Oct 14:95:117503.
CAS Number
– 2734916-64-2
Molecular Weight
– 339.43
SMILES
– C12=NC=CC=C1C(C3=CCN(CC4=CC=C5C=CC=CC5=C4)CC3)=CN2
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– ERK
Isoform
– ERK
Pathway
– MAPK/ERK Pathway;Stem Cell/Wnt
Product type
– Reference compound
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