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EN40
SKU
HY-122577-10 mg
Category Reference compound
Tags Aldehyde Dehydrogenase (ALDH), Cancer, Metabolic Enzyme/Protease
$450 – $3,350
Products Details
Product Description
– EN40 is a potent, selective aldehyde dehydrogenase 3A1 (ALDH3A1) inhibitor as a covalent ligand, exhibits an IC50 value of 2 uM[1]
Web ID
– HY-122577
Storage Temperature
– 4°C (Powder, stored under nitrogen)
Shipping
– Room Temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C13H15NO2
References
– [1]Counihan JL,et al.Chemoproteomics-Enabled Covalent Ligand Screening Reveals ALDH3A1 as a Lung Cancer Therapy Target.ACS Chem Biol. 2018 Aug 17;13(8):1970-1977
CAS Number
– 2094547-67-6
Molecular Weight
– 217.26
Compound Purity
– 99.56
SMILES
– C=CC(N1CCC(C)=C(C2=CC=CO2)C1)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : ≥ 100 mg/mL|Ethanol : 100 mg/mL (ultrasonic)
Target
– Aldehyde Dehydrogenase (ALDH)
Isoform
– ALDH3
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.