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EEDi-5273
$950 – $2,200
Products Details
Product Description
– EEDi-5273 is an exceptionally potent and orally efficacious EED inhibitor (IC50 = 0.2 nM) capable of achieving complete and persistent tumor regression.
Web ID
– HY-132922
Storage Temperature
– -20°C, 3 years (Powder)
Shipping
– Blue Ice
Applications
– Cancer-programmed cell death
Molecular Formula
– C26H22F4N6O2
References
– [1]Rej RK, et al. Discovery of EEDi-5273 as an Exceptionally Potent and Orally Efficacious EED Inhibitor Capable of Achieving Complete and Persistent Tumor Regression. J Med Chem. 2021 Oct 14;64(19):14540-14556.
CAS Number
– 2585648-55-9
Molecular Weight
– 526.49
Compound Purity
– 98.01
SMILES
– CC(N1CC2=CC(C(F)(F)F)=NC=C2C3=CN=C(N4C=NC(C1=O)=C34)NCC5=C6CCOC6=CC=C5F)C
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 25 mg/mL (ultrasonic)
Target
– Histone Methyltransferase
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
