Download Files:
(E/Z)-IT-603
Price range: 86 CAD through 2,928 CAD
Products Details
Product Description
– (E/Z)-IT-603 is a cell-permeable c-Rel inhibitor (IC50: 3μM) that directly and reversibly binds to c-Rel, altering its conformation and inhibiting its DNA binding and transcriptional activity.
Web ID
– T8799
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C11H9BrN2O3S
References
– Shono Y , Tuckett A Z , Ouk S , et al. A Small-Molecule c-Rel Inhibitor Reduces Alloactivation of T Cells without Compromising Antitumor Activity[J]. Cancer Discovery, 2014, 4(5):578-91.
CAS Number
– 292168-90-2
Molecular Weight
– C11H9BrN2O3S
Compound Purity
– 0.9897
SMILES
– COc1cc(Br)cc(C=C2NC(=S)NC2=O)c1O
Pathway
– NF-κB
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
Related Products
1000 in stock
1000 in stock
