Download Files:
dBRD4-BD1
Price range: 3,392 CAD through 5,920 CAD
For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.
Products Details
Product Description
– dBRD4-BD1 is a selective BRD4 bromodomain inhibitor. dBRD4-BD1 can selectively degrade BRD4 (DC50 = 280 nM). Notably, dBRD4-BD1 upregulates BRD2/3, a result not observed with degraders using pan-BET ligands. Designing BRD4 selectivity up front enables analysis of BRD4 biology without wider BET-inhibition and simplifies designing BRD4-selective heterobifunctional molecules, such as degraders with new E3 recruiting ligands or for additional probes beyond degraders.
Web ID
– T69506
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C50H53F3N8O9
CAS Number
– 2839318-19-1
Molecular Weight
– C50H53F3N8O9
SMILES
– O(C=1N=C(C2=C(N=CN2C3CCN(CCOCCOCCNC(COC4=C5C(C(=O)N(C5=O)C6C(=O)NC(=O)CC6)=CC=C4)=O)CC3)C7=CC=C(C(F)(F)F)C=C7)C=CN1)C8=CC(C(C)C)=CC=C8C
Pathway
– Others
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
Related Products
CDK ligand for PROTAC hydrochloride
Price range: 498 CAD through 3,170 CAD
1000 in stock
