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CDK12-IN-6
1,552 CAD
Only 1000 item(s) left in stock.
Products Details
Product Description
– CDK12-IN-6, a pyrazolotriazine compound, is a powerful inhibitor of CDK12. Its inhibitory activity is significant with an IC50 value of 1.19 μM when tested at high ATP concentration (2 mM). Notably, CDK12-IN-6 does not exhibit any inhibitory effect on CDK2/Cyclin E (IC50 >20 μM) and CDK9/Cyclin T1 (IC50 >20 μM) when tested under the same high ATP conditions (2 mM) (WO2021116178A1).
Web ID
– T40289
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C20H21F2N9
References
– Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.
CAS Number
– 2651196-71-1
Molecular Weight
– C20H21F2N9
SMILES
– Fc1ccc2nc(CNc3nc(nc4c(cnn34)C3CC3)N3CCNCC3)[nH]c2c1F
Pathway
– Others
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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