CDK12-IN-4
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CDK12-IN-4

SKU T40288-5 mg Category Brand:

1,552 CAD

Only 1000 item(s) left in stock.

Products Details

Product Description

– CDK12-IN-4, a pyrazolotriazine compound, exhibits potent inhibition of CDK12 by achieving an IC50 value of 0.641 μM, utilizing high ATP levels (2 mM). Notably, CDK12-IN-4 does not impact CDK2/Cyclin E (IC50 > 20 μM) or CDK9/Cyclin T1 (IC50 > 20 μM) under the influence of high ATP (2 mM) levels (WO2021116178A1).

Web ID

– T40288

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C20H20F2N8O

References

– Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.

CAS Number

– 2651196-69-7

Molecular Weight

– C20H20F2N8O

SMILES

– Fc1ccc2nc(CNc3nc(nc4c(cnn34)C3CC3)N3CCOCC3)[nH]c2c1F

Pathway

– Others

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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