Download Files:
CCG215022
Price range: 147 CAD through 2,608 CAD
Products Details
Product Description
– CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM for GRK2, 0.38±0.06 μM for GRK5, and 3.9±1 μM for GRK1.
Web ID
– T3498
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C26H22FN7O3
References
– Homan KT, et al. Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally DesignedInhibitor. J Biol Chem. 2015 Aug 21;290(34):20649-59.
CAS Number
– 1813527-81-9
Molecular Weight
– C26H22FN7O3
Compound Purity
– 0.9763
SMILES
– CC1=C(C(NC(=O)N1)c1ccc(F)c(c1)C(=O)NCc1ccccn1)C(=O)Nc1ccc2[nH]ncc2c1
Target
– Nucleoside Antimetabolite/Analog
Pathway
– Tyrosine Kinase/Adaptors|||GPCR/G Protein
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
Related Products
1000 in stock
1000 in stock
1000 in stock
