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Brilanestrant
Price range: 77 CAD through 1,035 CAD
Products Details
Product Description
– Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).
Web ID
– T5118
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C26H20ClFN2O2
Citations
– 1. Gao X, Ren X, Wang F, et al.Immunotherapy and drug sensitivity predictive roles of a novel prognostic model in hepatocellular carcinoma.Scientific Reports.2024, 14(1): 9509.
2. Yan X, Luo C, Yang J, et al.Antiviral Activity of Selective Estrogen Receptor Modulators against Severe Fever with Thrombocytopenia Syndrome Virus In Vitro and In Vivo.Viruses.2024, 16(8): 1332.
References
– By Lai, et al. Identification of GDC-0810 (ARN-810), an Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) that Demonstrates Robust Activity in Tamoxifen-Resistant Breast Cancer Xenografts. J Med Chem. 2015 Jun 25;58(12):4888-904.
CAS Number
– 1365888-06-7
Molecular Weight
– C26H20ClFN2O2
Compound Purity
– 0.9907
SMILES
– CCC(=C(c1ccc(C=CC(O)=O)cc1)c1ccc2[nH]ncc2c1)c1ccc(F)cc1Cl
Pathway
– Endocrinology/Hormones
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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