Download Files:
Products Details
Product Description
– BRD4 Inhibitor-17 (Compound 5i) is a potent inhibitor of BRD4 with an IC50 of 0.33 μM. BRD4 Inhibitor-17 plays crucial role in regulating transcription of inflammatory, proliferation and cell cycle genes. BRD4 Inhibitor-17 serves as potential antidotes for arsenicals[1].
Web ID
– HY-145909
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C16H16FN3O3S
References
– [1]Yatchang MF, et al. Development of BRD4 inhibitors as anti-inflammatory agents and antidotes for arsenicals. Bioorg Med Chem Lett. 2022;64:128696.
CAS Number
– 2835555-10-5
Molecular Weight
– 349.38
SMILES
– CC1=CC(S(=O)(NC2=CC3=C(NC(N(C3)C)=O)C=C2)=O)=CC=C1F
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
