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Apimostinel
$450 – $3,760
Products Details
Product Description
– Apimostinel (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist[1].
Web ID
– HY-102053
Storage Temperature
– 4°C (Powder, stored under nitrogen)
Shipping
– Room Temperature
Applications
– Neuroscience-Neurodegeneration
Molecular Formula
– C25H37N5O6
References
– [1]Naurex’s First Orally Active Molecule, NRX-1074, Demonstrates Statistically Significant Improvement in Depression Scores within 24 Hours in Phase 2 Study for Major Depressive Disorder. January 28, 2015.
CAS Number
– 1421866-48-9
Molecular Weight
– 503.59
Compound Purity
– 99.04
SMILES
– C[C@@H](O)[C@@H](C(N)=O)NC([C@@]1(CC2=CC=CC=C2)N(C([C@H]3N(C([C@H]([C@H](O)C)N)=O)CCC3)=O)CCC1)=O
Clinical Information
– Phase 1
Research Area
– Neurological Disease
Solubility
– DMSO : 155 mg/mL (ultrasonic)|H2O : ≥ 6.67 mg/mL
Target
– iGluR
Isoform
– NMDA Receptor
Pathway
– Membrane Transporter/Ion Channel;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
