![](https://immunomart.com/wp-content/uploads/2024/03/HY-149873.gif)
Download Files:
Anticancer agent 126
SKU
HY-149873-Get quote
Category Reference compound
Tags Cancer, Epigenetics, Histone Methyltransferase
Products Details
Product Description
– Anticancer agent 126 (compound 12) is a WDR5 inhibitor with anticancer effects. Anticancer agent 126 disrupts WDR5-MYC interaction in cells and reduce MYC target gene expression[1].
Web ID
– HY-149873
Shipping
– Room temperature
Molecular Formula
– C25H18F3N3O4S
References
– [1]Jian Ding, et al. Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC Interaction. J Med Chem. 2023 Jun 22;66(12):8310-8323.
Molecular Weight
– 513.49
SMILES
– FC1=C(C(F)=CC(C2=CC(S(=O)(F)=O)=CC=C2)=C1)CNC(C3=NN(C(C)=CC3=O)C4=CC=CC=C4)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Histone Methyltransferase
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.