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AHR antagonist 5 (free base)
SKU
HY-141609-1 mg
Category Reference compound
Tags Aryl Hydrocarbon Receptor, Cancer, Immunology/Inflammation
$190 – $1,200
Products Details
Product Description
– AHR antagonist 5 free base is a selective and orally active aryl hydrocarbon receptor (AHR) inhibitor. AHR antagonist 5 free base effectively blocks AHR from translocating from the cytoplasm to the nucleus. AHR antagonist 5 free base is highly selective for AHR over other receptors, transporters, and kinases[1].
Web ID
– HY-141609
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Applications
– Cancer-Kinase/protease
Molecular Formula
– C25H24FN7
References
– [1]Marta Sanchez-Martin, et al. Ahr inhibitors and uses thereof. WO2021142180A1.
CAS Number
– 2247950-42-9
Molecular Weight
– 441.50
Compound Purity
– 99.56
SMILES
– CC(C)C(C=N1)=C2N1C(N[C@H]3CC4=C(CC3)NC5=CC=CC=C45)=NC(C6=CN=CC(F)=C6)=N2
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– Aryl Hydrocarbon Receptor
Pathway
– Immunology/Inflammation
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.