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Products Details
Product Description
– AA10 is a potent and irreversible transglutaminase 2 (TG2) inhibitor for cancer research[1].
Web ID
– HY-157254
Shipping
– Room temperature
Molecular Formula
– C32H36N4O5
References
– [1]Akbar A, et al. Structure-Activity Relationships of Potent, Targeted Covalent Inhibitors That Abolish Both the Transamidation and GTP Binding Activities of Human Tissue Transglutaminase. J Med Chem. 2017 Sep 28;60(18):7910-7927.
CAS Number
– 2134106-02-6
Molecular Weight
– 556.65
SMILES
– O=C(OCC1=CC=CC=C1)N[C@H](C(N2CCN(C(C3=CC=C4C=CC=CC4=C3)=O)CC2)=O)CCCCNC(C=C)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Glutaminase
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
