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4-Me-PDTic HCl
Price range: 2,672 CAD through 4,480 CAD
Products Details
Product Description
– 4-Me-PDTic is a potent and selective Kappa Opioid Receptor Antagonist. 4-Me-PDTic had a Ke = 0.37 nM in a [35S]GTPγS binding assay and was 645- and >8100-fold selective for the κ relative to the μ and δ opioid receptors, respectively. Calculated logBB and CNS (central nervous system) multiparameter optimization (MPO) and low molecular weight values all predict that 4-Me-PDTic will penetrate the brain and pharmacokinetic studies in rats shows that 4-Me-PDTic does indeed penetrate the brain.
Web ID
– T69798
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C21H35Cl2N3O2
CAS Number
– 2209073-52-7
Molecular Weight
– C21H35Cl2N3O2
SMILES
– Cl.Cl.CC(C)[C@H](CN1CCC(C)CC1)NC(=O)[C@H]1Cc2ccc(O)cc2CN1
Pathway
– Others
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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