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Products Details
Product Description
– PROTAC ERα Degrader-4, a highly potent and selective agent (K i: 5.08 μM), contains OBHSAs, a linker, and E3 ligase ligands. This compound demonstrates superb inhibitory effects and ERα degradation activity in both Tamoxifen-sensitive and -resistant ER+ breast cancer (BC) cells, as well as in ERα-mutated BC cells. Additionally, PROTAC ERα Degrader-4 can induce apoptosis, making it valuable for cancer research.
Web ID
– T87263
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C55H62F3N5O10S2
CAS Number
– 2521299-80-7
Molecular Weight
– C55H62F3N5O10S2
SMILES
– S(N(CC(F)(F)F)C1=CC=C(OCCCCCC(N[C@H](C(=O)N2[C@H](C(N[C@@H](C)C3=CC=C(C=C3)C=4SC=NC4C)=O)C[C@@H](O)C2)C(C)(C)C)=O)C=C1)(=O)(=O)C5C6(C(=C(C(O6)(C5)[H])C7=CC=C(O)C=C7)C8=CC=C(O)C=C8)[H]
Product type
– PROTAC
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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