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PERK-IN-3
Price range: 2,672 CAD through 4,480 CAD
Products Details
Product Description
– PERK-IN-3 is a potent inhibitor of PERK (IC50 of 7.4 nM).
Web ID
– T12410
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C22H16F2N4O2
References
– Axten JM , et al. Discovery of 7-methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (GSK2606414), a potent and selective first-in-class inhibitor of protein kinase R (PKR)-like endoplasmic reticulum kinase (PERK). J Med Chem. 2012 Aug 23;55(16):7193-207.
CAS Number
– 1337532-08-7
Molecular Weight
– C22H16F2N4O2
SMILES
– NC1=C2C(=COC2=NC=N1)C=3C=C4C(=CC3)N(C(CC5=C(F)C=CC(F)=C5)=O)CC4
Target
– Epigenetic Reader Domain|||Ligands for Target Protein for PROTAC
Pathway
– MAPK
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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