L-803087

SKU T11800-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 48 CAD through 3,136 CAD

Products Details

Product Description

– L-803087 is a potent and selective agonist of the growth inhibitor sst4 receptor with a Ki value of 0.7 nM for sst4, demonstrating over 280-fold selectivity compared to other growth inhibitory receptors. L-803087 induces AMPA-mediated synaptic responses in the hippocampus in vitro and increases seizures in alginate-induced seizure-busting mice in vivo.

Web ID

– T11800

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C25H29F2N5O3

References

– Moneta D, et al. Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice. Eur J Neurosci. 2002 Sep;16(5):843-9.

CAS Number

– 217480-26-7

Molecular Weight

– C25H29F2N5O3

Compound Purity

– 0.9758

SMILES

– COC(=O)[C@H](CCCNC(N)=N)NC(=O)CCCc1c([nH]c2c(F)cc(F)cc12)-c1ccccc1

Target

– PROTAC Linker

Pathway

– GPCR/G Protein

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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