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GNA002
1,904 CAD
Only 1000 item(s) left in stock.
For Research Use Only (RUO). This product is sold strictly for laboratory research use. Not for human or veterinary consumption, therapeutic, or diagnostic use.
Products Details
Product Description
– GNA002 is a highly potent, specific, and covalent EZH2 (Enhancer of zeste homolog 2) inhibitor with an IC50 of 1.1 μM.
Web ID
– T11436
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C42H55NO8
References
– Wang X, et al. A covalently bound inhibitor triggers EZH2 degradation through CHIP-mediated ubiquitination. EMBO J. 2017 May, 36(9):1243-1260.
CAS Number
– 1385035-79-9
Molecular Weight
– C42H55NO8
SMILES
– [H][C@@]12C[C@@]3([H])C=C4C(=O)c5c(O)c(CC=C(/C)CCC=C(C)C)c(O)c(CC=C(C)C)c5O[C@@]14[C@@](CC=C(C)C(=O)NCCOCC)(OC2(C)C)C3=O
Target
– CFTR|||Autophagy
Pathway
– Chromatin/Epigenetic
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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