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Antihistamine-1
Price range: 85 CAD through 563 CAD
Products Details
Product Description
– Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).
Web ID
– T10335
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C23H24FN5
References
– Lavrador-Erb K, et al. The discovery and structure-activity relationships of 2-(piperidin-3-yl)-1H-benzimidazoles as selective, CNS penetrating H1-antihistamines for insomnia. Bioorg Med Chem Lett. 2010 May 1;20(9):2916-9.
CAS Number
– 1186430-60-3
Molecular Weight
– C23H24FN5
Compound Purity
– 1
SMILES
– C(N1C(=NC=2C1=CC=CC2)N3CCC(CC3)N4C=C(C)C=N4)C5=CC=C(F)C=C5
Target
– Others
Pathway
– Metabolism
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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