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Products Details
Product Description
– ZK168281 is a 25-carboxylic ester 1α,25(OH)2D3 analog and a pure VDR antagonist (Kd of 0.1 nM), efficiently inhibiting the coactivator (CoA) interaction with its receptor.
Web ID
– T13404
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C32H46O5
References
– Lempiäinen H, et al. Antagonist- and inverse agonist-driven interactions of the vitamin D receptor and the constitutive androstane receptor with corepressor protein. Mol Endocrinol. 2005 Sep;19(9):2258-72.
CAS Number
– 186371-96-0
Molecular Weight
– C32H46O5
SMILES
– [H][C@@]12CC[C@H]([C@H](C)C=C[C@@H](O)C3(CC3)C=CC(=O)OCC)[C@@]1(C)CCCC2=C/C=C1/C[C@@H](O)C[C@H](O)C1=C
Target
– PDE
Pathway
– Others
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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