WDR5-0102

SKU T67947-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 112 CAD through 3,664 CAD

Products Details

Product Description

– WDR5-0102 is a compound that inhibits the WDR5-MLL1 interface (K dis = 7 μM, K d = 4 μM), selectively reducing MLL1 HMT activity without affecting the human H3K4 methyltransferase SETD7 or other HMTs, including G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5.

Web ID

– T67947

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C18H19ClN4O3

References

– Lawrence HR, et al. Inhibitors of Src homology-2 domain containing protein tyrosine phosphatase-2 (Shp2) based on oxindole scaffolds. J Med Chem. 2008;51(16):4948-4956.

CAS Number

– 824960-50-1

Molecular Weight

– C18H19ClN4O3

Compound Purity

– 0.9716

SMILES

– N(C(=O)C1=C(Cl)C=CC=C1)C2=C(C=CC(N(=O)=O)=C2)N3CCN(C)CC3

Pathway

– Chromatin/Epigenetic

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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