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Products Details
Product Description
– SOS1-IN-16 (Comp 54) is a selective inhibitor of SOS1 with an IC50 of 7.2 nM. SOS1-IN-16 has inhibitory activity of CYP3A4 when using testosterone as a substrate, with an IC50 of 8.9μM. SOS1-IN-16 can be used for cancer research[1].
Web ID
– HY-153989
Shipping
– Room temperature
Molecular Formula
– C30H31F3N4O3
References
– [1]Chen SJ, et.al.Polysubstituted benzazepine heteroaryl derivative and application thereof
CAS Number
– 2930763-85-0
Molecular Weight
– 552.59
SMILES
– C[C@H](C1=C(C(C(F)(F)CO)=CC=C1)F)NC2=NC(C)=NC3=C2C=C(C4=CC(CC(N(C)C)=O)=C(C=C4)OC)C=C3
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Cytochrome P450;Ras
Pathway
– GPCR/G Protein;Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
