Sigma-1 receptor antagonist 3
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Sigma-1 receptor antagonist 3

SKU T12912-1 mg Category Brand:

Price range: 130 CAD through 1,525 CAD

Products Details

Product Description

– Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 μM)

Web ID

– T12912

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C19H23ClFN3O

References

– Lan Y, et al. Synthesis and biological evaluation of novel sigma-1 receptor antagonists based on pyrimidine scaffold as agents for treating neuropathic pain. J Med Chem. 2014 Dec 26;57(24):10404-23.

CAS Number

– 1639220-17-9

Molecular Weight

– C19H23ClFN3O

Compound Purity

– 1

SMILES

– Cc1nc(nc(OCCCN2CCCCC2)c1Cl)-c1ccc(F)cc1

Target

– Others

Pathway

– GPCR/G Protein|||Membrane transporter/Ion channel

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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