Selpercatinib
Add to CompareAdded to Compare

Download Files:

Selpercatinib

SKU T8222-2 mg Category Brand:

Price range: 48 CAD through 1,840 CAD

Products Details

Product Description

– Selpercatinib (LOXO-292) is a tyrosine kinase inhibitor with antineoplastic properties, displaying IC50 values of 14.0 nM for RET (WT), 24.1 nM for RET (V804M), and 530.7 nM for RET (G810R).

Web ID

– T8222

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C29H31N7O3

Citations

– 1. Li S, Liu Z, Jiao X, et al.Selpercatinib attenuates bleomycin-induced pulmonary fibrosis by inhibiting the TGF-β1 signaling pathway.Biochemical Pharmacology.2024: 116282.

References

– Steven W. Andrews, et al. Substituted pyrazolo[1,5-a]pyridine compounds as ret kinase inhibitors. WO2018071447A1.

CAS Number

– 2152628-33-4

Molecular Weight

– C29H31N7O3

Compound Purity

– 0.9989

SMILES

– COc1ccc(CN2C3CC2CN(C3)c2ccc(cn2)-c2cc(OCC(C)(C)O)cn3ncc(C#N)c23)cn1

Pathway

– Apoptosis|||Tyrosine Kinase/Adaptors

Product type

– Small Compound

Booklet

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

Related Products

Select options
Mecarbinate
Mecarbinate Price range: 46 CAD through 56 CAD
1 g1 mL * 10 mM (in DMSO)

1000 in stock

Select options
Mephenesin
Mephenesin Price range: 53 CAD through 173 CAD
1 g10 g5 g

1000 in stock

Select options
Flubendazole
Flubendazole Price range: 53 CAD through 149 CAD
1 mL * 10 mM (in DMSO)100 mg50 mg

1000 in stock

Select options
Atenolol Hydrochloride
Atenolol Hydrochloride Price range: 2,432 CAD through 4,000 CAD
100 mg25 mg50 mg

1000 in stock

Select options
2,2'-Bipyridine
2,2′-Bipyridine Price range: 46 CAD through 171 CAD
1 g100 mg500 mg

1000 in stock

My Cart
Wishlist
Recently Viewed
Categories

Request Data Sheet / Safty Data Sheet

Please enable JavaScript in your browser to complete this form.
=

Price Request

Please enable JavaScript in your browser to complete this form.
=

Compare Products (0 Products)
document.addEventListener('elementor/popup/show', function() { if (typeof turnstile !== 'undefined') { document.querySelectorAll('.cf-turnstile').forEach(function(el) { if (!el.dataset.rendered) { turnstile.render(el); el.dataset.rendered = true; } }); } });