Samelisant

SKU T9770-1 mL * 10 mM (in DMSO) Category Brand:

Price range: 181 CAD through 4,624 CAD

Products Details

Product Description

– Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects and can be used in studies about narcolepsy.

Web ID

– T9770

Storage Temperature

– -20℃

Shipping

– Blue Ice

Molecular Formula

– C21H31N3O3

References

– Nirogi R, et al. Samelisant (SUVN-G3031), a potent, selective and orally active histamine H3 receptor inverse agonist for the potential treatment of narcolepsy: pharmacological and neurochemical characterisation. Psychopharmacology (Berl). 2021 Jun;238(6):1495-1511.

CAS Number

– 1394808-82-2

Molecular Weight

– C21H31N3O3

Compound Purity

– 0.9909

SMILES

– O(C1CCN(CC1)C2CCC2)C3=CC=C(NC(CN4CCOCC4)=O)C=C3

Pathway

– Neuroscience|||GPCR/G Protein|||Immunology/Inflammation

Product type

– Small Compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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