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PKC-theta inhibitor
$152 – $2,150
Products Details
Product Description
– PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM.
Web ID
– HY-112681
Storage Temperature
– -20°C, 3 years; 4°C, 2 years (Powder)
Shipping
– Room Temperature
Molecular Formula
– C20H25F3N6O3
References
– [1]Cywin CL, et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30.
CAS Number
– 736048-65-0
Molecular Weight
– 454.45
Compound Purity
– 99.37
SMILES
– FC(F)(F)OC1=CC=CC=C1CNC2=NC=C([N+]([O-])=O)C(NCC3CCC(CN)CC3)=N2
Clinical Information
– No Development Reported
Research Area
– Others
Solubility
– DMSO : 62.5 mg/mL (ultrasonic)
Target
– PKC
Isoform
– PKCθ
Pathway
– Epigenetics;TGF-beta/Smad
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
