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PD 151746
Price range: 94 CAD through 507 CAD
Products Details
Product Description
– PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 ± 0.03 μM) over m-calpain (Ki = 5.33 ± 0.77 μM). Its IC50 values are 0.26 ± 0.03 μM (Ki for μ-calpain) and 5.33 ± 0.77 μM (Ki for m-calpain) [1]. In vitro, PD151746 targets calpain and reduces oxLDL-induced cytotoxicity [2].
Web ID
– T2493
Storage Temperature
– -20℃
Shipping
– Blue Ice
Molecular Formula
– C11H8FNO2S
References
– Wang KK, et al. Proc Natl Acad Sci U S A. 1996, 93(13), 6687-6692.
CAS Number
– 179461-52-0
Molecular Weight
– C11H8FNO2S
Compound Purity
– 0.9863
SMILES
– OC(=O)C(S)=Cc1c[nH]c2ccc(F)cc12
Pathway
– Proteases/Proteasome|||Ubiquitination
Product type
– Small Compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
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